7SFO
Estrogen Receptor Alpha Ligand Binding Domain Y537S in Complex with 3-(((2-chloro-5-phenylthieno[2,3-d]pyrimidin-4-yl)amino)methyl)phenol and GRIP Peptide
Summary for 7SFO
Entry DOI | 10.2210/pdb7sfo/pdb |
Descriptor | Estrogen receptor, Nuclear receptor coactivator 2, 3-{[(2-chloro-5-phenylthieno[2,3-d]pyrimidin-4-yl)amino]methyl}phenol, ... (4 entities in total) |
Functional Keywords | estrogen receptor, hormone, breast cancer, alpha helical bundle, transcription |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 4 |
Total formula weight | 60169.69 |
Authors | Joyner, C.,Reddy, V.K.,Wilson, T.,Fanning, S.W. (deposition date: 2021-10-04, release date: 2022-10-12, Last modification date: 2023-10-18) |
Primary citation | Fanning, S.W. Estrogen Receptor Alpha To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
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