7Q10
Acetyltrasferase(3) type IIIa in complex with 3-N-methyl-nemycin B
Summary for 7Q10
Entry DOI | 10.2210/pdb7q10/pdb |
Related | 7Q0Q |
Descriptor | Aminoglycoside N(3)-acetyltransferase III, GLYCEROL, 3N methyl nemycin B, ... (7 entities in total) |
Functional Keywords | acetyltrasferase, aminoglycosides, inhibitor, complex, antibiotic |
Biological source | Pseudomonas aeruginosa |
Total number of polymer chains | 2 |
Total formula weight | 60474.41 |
Authors | Pontillo, N.,Guskov, A. (deposition date: 2021-10-17, release date: 2022-11-02, Last modification date: 2024-01-31) |
Primary citation | Pontillo, N.,Warszawik, E.M.,Partipilo, M.,Stetsenko, A.,Loznik, M.,Yang, X.,Slotboom, D.J.,Guskov, A.,Herrmann, A. 3-N-alkylation in aminoglycoside antibiotic neomycin B overcomes bacterial resistance mediated by acetyltransferase (3) IIIa To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.82 Å) |
Structure validation
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