7OOV
Crystal structure of PIM1 in complex with ARC-1411
Summary for 7OOV
Entry DOI | 10.2210/pdb7oov/pdb |
Related PRD ID | PRD_002337 |
Descriptor | Serine/threonine-protein kinase pim-1, Inhibitor ARC-1411, SULFATE ION, ... (5 entities in total) |
Functional Keywords | pim1, inhibitor, kinase, kinase substrate, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 37530.79 |
Authors | Chaikuad, A.,Dixon-Clarke, S.E.,Nonga, O.E.,Uri, A.,Bullock, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2021-05-28, release date: 2021-08-04, Last modification date: 2024-04-10) |
Primary citation | Nonga, O.E.,Lavogina, D.,Enkvist, E.,Kestav, K.,Chaikuad, A.,Dixon-Clarke, S.E.,Bullock, A.N.,Kopanchuk, S.,Ivan, T.,Ekambaram, R.,Viht, K.,Knapp, S.,Uri, A. Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM Family. Molecules, 26:-, 2021 Cited by PubMed: 34299628DOI: 10.3390/molecules26144353 PDB entries with the same primary citation |
Experimental method |
Structure validation
Download full validation report