7CRF
Crystal structure of human TLR8 in complex with CU-CPD107
Summary for 7CRF
Entry DOI | 10.2210/pdb7crf/pdb |
Descriptor | Toll-like receptor 8, alpha-D-mannopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (10 entities in total) |
Functional Keywords | immune system |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 196905.83 |
Authors | Sakaniwa, K.,Tanji, H.,Ohto, U.,Shimizu, T. (deposition date: 2020-08-13, release date: 2021-06-23, Last modification date: 2023-11-29) |
Primary citation | Yang, Y.,Csakai, A.,Jiang, S.,Smith, C.,Tanji, H.,Huang, J.,Jones, T.,Sakaniwa, K.,Broadwell, L.,Shi, C.,Soti, S.,Ohto, U.,Fang, Y.,Shen, S.,Deng, F.,Shimizu, T.,Yin, H. Tetrasubstituted imidazoles as incognito Toll-like receptor 8 a(nta)gonists. Nat Commun, 12:4351-4351, 2021 Cited by PubMed: 34272380DOI: 10.1038/s41467-021-24536-4 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.89 Å) |
Structure validation
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