7BCH
Notum Fragment 772
Summary for 7BCH
Entry DOI | 10.2210/pdb7bch/pdb |
Related | 7B84 |
Descriptor | Palmitoleoyl-protein carboxylesterase NOTUM, SULFATE ION, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (5 entities in total) |
Functional Keywords | notum inhibitor, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 44351.82 |
Authors | Zhao, Y.,Jones, E.Y. (deposition date: 2020-12-19, release date: 2022-01-12, Last modification date: 2024-10-16) |
Primary citation | Zhao, Y.,Mahy, W.,Willis, N.J.,Woodward, H.L.,Steadman, D.,Bayle, E.D.,Atkinson, B.N.,Sipthorp, J.,Vecchia, L.,Ruza, R.R.,Harlos, K.,Jeganathan, F.,Constantinou, S.,Costa, A.,Kjaer, S.,Bictash, M.,Salinas, P.C.,Whiting, P.,Vincent, J.P.,Fish, P.V.,Jones, E.Y. Structural Analysis and Development of Notum Fragment Screening Hits. Acs Chem Neurosci, 13:2060-2077, 2022 Cited by PubMed: 35731924DOI: 10.1021/acschemneuro.2c00325 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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