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6ZCX

SYK Kinase domain in complex with azabenzimidazole inhibitor 18

Summary for 6ZCX
Entry DOI10.2210/pdb6zcx/pdb
DescriptorTyrosine-protein kinase SYK, ~{N},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{R})-piperidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamide (3 entities in total)
Functional Keywordssyk kinase transferase inhibitor, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight35341.50
Authors
Read, J.A. (deposition date: 2020-06-12, release date: 2021-06-23, Last modification date: 2024-01-24)
Primary citationRead, J.A.
SYK Kinase domain in complex with azabenzimidazole inhibitor 18
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.66 Å)
Structure validation

221051

數據於2024-06-12公開中

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