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6Z4Y

Crystal structure of Aurora A (STK6) in complex with macrocycle ODS2003208

Summary for 6Z4Y
Entry DOI10.2210/pdb6z4y/pdb
DescriptorAurora kinase A, CITRIC ACID, 1,2-ETHANEDIOL, ... (5 entities in total)
Functional Keywordskinase, kinase inhibitor, aurora a, stk6, macrocycle, nanocyclic, structural genomics, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight34083.86
Authors
Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2020-05-26, release date: 2020-06-03, Last modification date: 2024-01-24)
Primary citationChaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of Aurora A (STK6) in complex with macrocycle ODS2003208
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.25 Å)
Structure validation

221051

數據於2024-06-12公開中

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