6YNC
Crystal structure of cAMP-dependent Protein Kinase (PKA) in complex with the methylated Fasudil-derived fragment N-methylisoquinoline-5-sulfonamide (soaked)
6YNC の概要
エントリーDOI | 10.2210/pdb6ync/pdb |
分子名称 | cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha, ~{N}-methylisoquinoline-5-sulfonamide, ... (4 entities in total) |
機能のキーワード | phosphotransferase, signalling pathways, glycogen metabolism, serine/threonine kinase, transferase |
由来する生物種 | Cricetulus griseus (Chinese hamster) 詳細 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 43409.33 |
構造登録者 | Oebbeke, M.,Wienen-Schmidt, B.,Heine, A.,Klebe, G. (登録日: 2020-04-13, 公開日: 2020-10-14, 最終更新日: 2024-01-24) |
主引用文献 | Wienen-Schmidt, B.,Oebbeke, M.,Ngo, K.,Heine, A.,Klebe, G. Two Methods, One Goal: Structural Differences between Cocrystallization and Crystal Soaking to Discover Ligand Binding Poses. Chemmedchem, 16:292-300, 2021 Cited by PubMed: 33029876DOI: 10.1002/cmdc.202000565 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.4 Å) |
構造検証レポート
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