6UMD

Crystal structure of human GAC in complex with inhibitor UPGL00012

6UMD の概要

• エントリーDOI: 10.2210/pdb6umd/pdb
• 分子名称: Glutaminase kidney isoform, mitochondrial, 2-(pyridin-3-yl)-N-(5-{4-[(5-{[(pyridin-3-yl)acetyl]amino}-1,3,4-thiadiazol-2-yl)amino]piperidin-1-yl}-1,3,4-thiadiazol-2-yl)acetamide (3 entities in total)
• 機能のキーワード: inhibitor, complex, hydrolase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
• 由来する生物種: Homo sapiens (Human)
• タンパク質・核酸の鎖数: 4
• 化学式量合計: 233281.44

構造登録者

Huang, Q.,Cerione, R.A. (登録日: 2019-10-09, 公開日: 2020-10-14, 最終更新日: 2023-10-11)

• 主引用文献: Huang, Q.,Cerione, R.A.; Crystal structure of human GAC in complex with inhibitor UPGL00012; To Be Published,

実験手法

X-RAY DIFFRACTION (2.7 Å)