6TW8
Leishmania major N-myristoyltransferase in complex with indazole inhibitor IMP-917
This is a non-PDB format compatible entry.
Summary for 6TW8
Entry DOI | 10.2210/pdb6tw8/pdb |
Related | 5O6H |
Descriptor | Glycylpeptide N-tetradecanoyltransferase, TETRADECANOYL-COA, 1-[5-[4-fluoranyl-2-[2-(1,3,5-trimethylpyrazol-4-yl)ethoxy]phenyl]-2~{H}-indazol-3-yl]-~{N},~{N}-dimethyl-methanamine, ... (5 entities in total) |
Functional Keywords | transferase, myristoylation, indazole, leishmania |
Biological source | Leishmania major |
Total number of polymer chains | 2 |
Total formula weight | 99238.95 |
Authors | Brannigan, J.A. (deposition date: 2020-01-12, release date: 2021-07-21, Last modification date: 2024-05-15) |
Primary citation | Brannigan, J.A. Leishmania major N-myristoyltransferase in complex with indazole inhibitor IMP-917 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.79 Å) |
Structure validation
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