6TRY
Crystal structure of human Aldehyde dehydrogenase 1A3 in complex with MF13 inhibitor compound
6TRY の概要
エントリーDOI | 10.2210/pdb6try/pdb |
分子名称 | Aldehyde dehydrogenase family 1 member A3, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, 8-(4-chlorophenyl)-2-phenyl-imidazo[1,2-a]pyridine, ... (5 entities in total) |
機能のキーワード | dehydrogenase isoenzyme aldh1a3 selective inhibitor high grade glioma, oxidoreductase |
由来する生物種 | Homo sapiens (Human) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 114383.07 |
構造登録者 | |
主引用文献 | Quattrini, L.,Gelardi, E.L.M.,Petrarolo, G.,Colombo, G.,Ferraris, D.M.,Picarazzi, F.,Rizzi, M.,Garavaglia, S.,La Motta, C. Progress in the Field of Aldehyde Dehydrogenase Inhibitors: Novel Imidazo[1,2- a ]pyridines against the 1A Family. Acs Med.Chem.Lett., 11:963-970, 2020 Cited by PubMed: 32435412DOI: 10.1021/acsmedchemlett.9b00686 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.9 Å) |
構造検証レポート
検証レポート(詳細版)
をダウンロード
![ダウンロード](/newweb/media/icons/dl.png)