6T9R
Aplysia californica AChBP in complex with a cytisine derivative
This is a non-PDB format compatible entry.
Summary for 6T9R
Entry DOI | 10.2210/pdb6t9r/pdb |
Descriptor | Acetylcholine binding protein, (1~{R},9~{S})-5-(3-oxidanylpropyl)-7,11-diazatricyclo[7.3.1.0^{2,7}]trideca-2,4-dien-6-one, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (8 entities in total) |
Functional Keywords | acetylcholine binding protein, nicotinic receptor surrogate, hydrolase |
Biological source | Aplysia californica (California sea hare) |
Total number of polymer chains | 10 |
Total formula weight | 293433.86 |
Authors | Davis, S.,Hunter, W.N. (deposition date: 2019-10-28, release date: 2020-02-12, Last modification date: 2024-01-24) |
Primary citation | Davis, S.,Rego Campello, H.,Gallagher, T.,Hunter, W.N. The thermodynamic profile and molecular interactions of a C(9)-cytisine derivative-binding acetylcholine-binding protein from Aplysia californica. Acta Crystallogr.,Sect.F, 76:74-80, 2020 Cited by PubMed: 32039888DOI: 10.1107/S2053230X20001168 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.72 Å) |
Structure validation
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