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6RMY

Human Carbonic anhydrase II mutant T199V bound by 3-(cyclooctylamino)-2,5,6-trifluoro-4-[(2-hydroxyethyl)sulfonyl]benzenesulfonamide

Summary for 6RMY
Entry DOI10.2210/pdb6rmy/pdb
DescriptorCarbonic anhydrase 2, ZINC ION, 3-(cyclooctylamino)-2,5,6-trifluoro-4-[(2-hydroxyethyl)sulfonyl]benzenesulfonamide, ... (7 entities in total)
Functional Keywordsdrug design, carbonic anhydrase, benzenesulfonamide, metal-binding, lyase-lyase inhibitor complex, lyase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight30233.53
Authors
Smirnov, A.,Paketuryte, V.,Manakova, E.,Grazulis, S. (deposition date: 2019-05-07, release date: 2020-06-03, Last modification date: 2024-01-24)
Primary citationSmirnov, A.,Manakova, E.,Grazulis, S.,Paketuryte, V.
Human Carbonic anhydrase II mutant T199V bound by 3-(cyclooctylamino)-2,5,6-trifluoro-4-[(2-hydroxyethyl)sulfonyl]benzenesulfonamide
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

220472

数据于2024-05-29公开中

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