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6PZP

Crystal structure of caspase-1 in complex with VX-765

Summary for 6PZP
Entry DOI10.2210/pdb6pzp/pdb
DescriptorCaspase-1, N-(4-amino-3-chlorobenzene-1-carbonyl)-3-methyl-L-valyl-N-[(2S)-1-carboxy-3-oxopropan-2-yl]-L-prolinamide, ... (4 entities in total)
Functional Keywordsprotease, complex, inhibitor, immune system
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight30609.53
Authors
Yang, J.,Liu, Z.,Xiao, T.S. (deposition date: 2019-08-01, release date: 2020-08-05, Last modification date: 2023-10-11)
Primary citationYang, J.,Liu, Z.,Xiao, T.S.
Crystal structure of caspase-1 in complex with VX-765
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.94 Å)
Structure validation

221051

數據於2024-06-12公開中

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