6PG8
WDR5delta23 bound to (2-(3-phenylpropyl)-1H-imidazol-4-yl)methanol
Summary for 6PG8
Entry DOI | 10.2210/pdb6pg8/pdb |
Related | 6PG3 |
Descriptor | WD repeat-containing protein 5, [2-(3-phenylpropyl)-1H-imidazol-4-yl]methanol, CHLORIDE ION, ... (5 entities in total) |
Functional Keywords | inhibitor, scaffolding protein, b-propellor, chromatin regulator, protein binding, protein binding-inhibitor complex, protein binding/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 138895.18 |
Authors | Dennis, M.L.,Peat, T.S. (deposition date: 2019-06-24, release date: 2019-12-11, Last modification date: 2023-10-11) |
Primary citation | Dennis, M.L.,Morrow, B.J.,Dolezal, O.,Cuzzupe, A.N.,Stupple, A.E.,Newman, J.,Bentley, J.,Hattarki, M.,Nuttall, S.D.,Foitzik, R.C.,Street, I.P.,Stupple, P.A.,Monahan, B.J.,Peat, T.S. Fragment screening for a protein-protein interaction inhibitor to WDR5. Struct Dyn., 6:064701-064701, 2019 Cited by PubMed: 31768400DOI: 10.1063/1.5122849 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.67 Å) |
Structure validation
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