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6K1Q

Human endothelin receptor type-B in complex with inverse agonist IRL2500

Summary for 6K1Q
Entry DOI10.2210/pdb6k1q/pdb
DescriptorEndothelin B receptor,Endolysin,Endothelin B receptor, (2~{S})-2-[[(2~{R})-2-[(3,5-dimethylphenyl)carbonyl-methyl-amino]-3-(4-phenylphenyl)propanoyl]amino]-3-(1~{H}-indol-3-yl)propanoic acid, PHOSPHATE ION, ... (5 entities in total)
Functional Keywordsalpha helical, signaling protein
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains1
Total formula weight55933.97
Authors
Nagiri, C.,Shihoya, W.,Nureki, O. (deposition date: 2019-05-11, release date: 2019-07-17)
Primary citationNagiri, C.,Shihoya, W.,Inoue, A.,Kadji, F.M.N.,Aoki, J.,Nureki, O.
Crystal structure of human endothelin ETBreceptor in complex with peptide inverse agonist IRL2500.
Commun Biol, 2:236-236, 2019
Cited by
PubMed: 31263780
DOI: 10.1038/s42003-019-0482-7
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.7 Å)
Structure validation

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