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6JJ5

BRD4 in complex with 259

Summary for 6JJ5
Entry DOI10.2210/pdb6jj5/pdb
DescriptorBromodomain-containing protein 4, 3-((1-methyl-2-oxo-1,2,2a1,5a-tetrahydro-6H-pyrido[3',2':6,7]azepino[4,3,2-cd]isoindol-6-yl)methyl)benzamide (3 entities in total)
Functional Keywordsbrd4, inhibitor, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15265.60
Authors
Xu, J.,Chen, Y.,Jiang, F.,Zhu, J. (deposition date: 2019-02-25, release date: 2020-02-26, Last modification date: 2024-03-27)
Primary citationXu, J.,Zhu, J.,Chen, Y.,Jiang, F.
BRD4 in complex with ZZM1
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.2 Å)
Structure validation

218500

數據於2024-04-17公開中

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