6JI4

brd4-bd1 bound with ligand 138

Summary for 6JI4

• Entry DOI: 10.2210/pdb6ji4/pdb
• Descriptor: Bromodomain-containing protein 4, (3R)-4-cyclopropyl-1,3-dimethyl-6-[5-methyl-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]-3,4-dihydroquinoxalin-2(1H)-one (3 entities in total)
• Functional Keywords: dna damage, transcription regulation, bromodomain-containing protein 4, transcription
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 15010.36

Authors

Cao, D.Y.,Li, Y.L.,Du, Z.Y.,Li, J.,Xiong, B. (deposition date: 2019-02-20, release date: 2020-02-26, Last modification date: 2023-11-22)

• Primary citation: Cao, D.Y.,Li, Y.L.,Du, Z.Y.,Li, J.,Xiong, B.; brd4-bd1 bound with ligand 138; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.6 Å)