6IIN
USP14 catalytic domain with IU1-248
Summary for 6IIN
Entry DOI | 10.2210/pdb6iin/pdb |
Descriptor | Ubiquitin carboxyl-terminal hydrolase 14, 4-{3-[(4-hydroxypiperidin-1-yl)acetyl]-2,5-dimethyl-1H-pyrrol-1-yl}benzonitrile (3 entities in total) |
Functional Keywords | usp14 inhibitor complex, structural protein, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 88733.07 |
Authors | Mei, Z.Q.,Wang, J.W.,Wang, F.,Wang, Y.W. (deposition date: 2018-10-07, release date: 2018-12-19, Last modification date: 2024-03-27) |
Primary citation | Wang, Y.,Jiang, Y.,Ding, S.,Li, J.,Song, N.,Ren, Y.,Hong, D.,Wu, C.,Li, B.,Wang, F.,He, W.,Wang, J.,Mei, Z. Small molecule inhibitors reveal allosteric regulation of USP14 via steric blockade. Cell Res., 28:1186-1194, 2018 Cited by PubMed: 30254335DOI: 10.1038/s41422-018-0091-x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.53 Å) |
Structure validation
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