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6HKX

Eg5-inhibitor complex

Summary for 6HKX
Entry DOI10.2210/pdb6hkx/pdb
DescriptorKinesin-like protein KIF11, ADENOSINE-5'-DIPHOSPHATE, (2~{S})-2-(3-azanylpropyl)-5-[2,5-bis(fluoranyl)phenyl]-~{N}-methoxy-~{N}-methyl-2-phenyl-1,3,4-thiadiazole-3-carboxamide, ... (6 entities in total)
Functional Keywordseg5, kif11, eg5-inhibitor, cell cycle
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight84067.37
Authors
Talapatra, S.K.,Kozielski, F. (deposition date: 2018-09-09, release date: 2019-09-25, Last modification date: 2024-01-17)
Primary citationIndorato, R.L.,Talapatra, S.K.,Lin, F.,Haider, S.,Mackay, S.P.,Kozielski, F.,Skoufias, D.A.
Is the Fate of Clinical Candidate Arry-520 Already Sealed? Predicting Resistance in Eg5-Inhibitor Complexes.
Mol.Cancer Ther., 18:2394-2406, 2019
Cited by
PubMed: 31488701
DOI: 10.1158/1535-7163.MCT-19-0154
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.8 Å)
Structure validation

217157

건을2024-03-13부터공개중

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