6GHK
Human PARP1 (ARTD1) - Catalytic domain in complex with inhibitor ME0527
Summary for 6GHK
Entry DOI | 10.2210/pdb6ghk/pdb |
Descriptor | Poly [ADP-ribose] polymerase 1, ~{N}-[(1~{R})-1-(4-imidazol-1-ylphenyl)ethyl]-3-(4-oxidanylidene-1~{H}-quinazolin-2-yl)propanamide, SULFATE ION, ... (4 entities in total) |
Functional Keywords | inhibitor, adp-ribosyl transferase, protein-ligand complex, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 81751.14 |
Authors | Karlberg, T.,Thorsell, A.G.,Lindgren, A.E.G.,Moche, M.,Brock, J.,Ekblad, T.,Spjut, S.,Elofsson, M.,Schuler, H. (deposition date: 2018-05-08, release date: 2019-05-22, Last modification date: 2024-01-17) |
Primary citation | Karlberg, T.,Thorsell, A.G.,Lindgren, A.E.G.,Ekblad, T.,Spjut, S.,Elofsson, M.,Schuler, H. Human PARP1 (ARTD1) - Catalytic domain in complex with inhibitor ME0527 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.28 Å) |
Structure validation
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