6FZP
PPAR gamma complex.
Summary for 6FZP
Entry DOI | 10.2210/pdb6fzp/pdb |
Descriptor | Peroxisome proliferator-activated receptor gamma, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, (2~{S})-3-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]phenyl]-2-[[2-(phenylcarbonyl)phenyl]amino]propanoic acid, ... (4 entities in total) |
Functional Keywords | nuclear receptor, transcription |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 33468.94 |
Authors | Rochel, N.,Beji, S. (deposition date: 2018-03-15, release date: 2019-02-13, Last modification date: 2024-01-17) |
Primary citation | Rochel, N.,Krucker, C.,Coutos-Thevenot, L.,Osz, J.,Zhang, R.,Guyon, E.,Zita, W.,Vanthong, S.,Hernandez, O.A.,Bourguet, M.,Badawy, K.A.,Dufour, F.,Peluso-Iltis, C.,Heckler-Beji, S.,Dejaegere, A.,Kamoun, A.,de Reynies, A.,Neuzillet, Y.,Rebouissou, S.,Beraud, C.,Lang, H.,Massfelder, T.,Allory, Y.,Cianferani, S.,Stote, R.H.,Radvanyi, F.,Bernard-Pierrot, I. Recurrent activating mutations of PPAR gamma associated with luminal bladder tumors. Nat Commun, 10:253-253, 2019 Cited by PubMed: 30651555DOI: 10.1038/s41467-018-08157-y PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
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