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6FMP

Keap1 - peptide complex

Summary for 6FMP
Entry DOI10.2210/pdb6fmp/pdb
DescriptorKelch-like ECH-associated protein 1, ACY-ASP-GLU-GLU-THR-GLY-GLU-PHE, ACETATE ION, ... (7 entities in total)
Functional Keywordskeap1, kelch-domain, nrf2, neurodegenerative, inhibitor, peptide binding protein
Biological sourceHomo sapiens (human)
More
Total number of polymer chains3
Total formula weight93640.06
Authors
Talapatra, S.K.,Kozielski, F.,Wells, G.,Georgakopoulos, N.D. (deposition date: 2018-02-01, release date: 2018-08-08, Last modification date: 2024-02-07)
Primary citationGeorgakopoulos, N.D.,Talapatra, S.K.,Gatliff, J.,Kozielski, F.,Wells, G.
Modified Peptide Inhibitors of the Keap1-Nrf2 Protein-Protein Interaction Incorporating Unnatural Amino Acids.
Chembiochem, 19:1810-1816, 2018
Cited by
PubMed: 29927029
DOI: 10.1002/cbic.201800170
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.92 Å)
Structure validation

218500

건을2024-04-17부터공개중

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