6BQP

Crystal Structure of the Human CAMKK2B in complex with Crenolanib

6BQP の概要

• エントリーDOI: 10.2210/pdb6bqp/pdb
• 分子名称: Calcium/calmodulin-dependent protein kinase kinase 2, 1-(2-{5-[(3-Methyloxetan-3-yl)methoxy]-1H-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amine, 1,2-ETHANEDIOL, ... (4 entities in total)
• 機能のキーワード: transferase, protein kinase domain, structural genomics, structural genomics consortium, sgc, transferase inhibitor complex
• 由来する生物種: Homo sapiens (Human)
• タンパク質・核酸の鎖数: 1
• 化学式量合計: 33632.86

構造登録者

Counago, R.M.,de Souza, G.P.,dos Reis, C.V.,Ramos, P.Z.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) (登録日: 2017-11-28, 公開日: 2017-12-13, 最終更新日: 2023-10-04)

• 主引用文献: Counago, R.M.,de Souza, G.P.,dos Reis, C.V.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC); Crystal Structure of the Human CAMKK2B in complex with Crenolanib; To Be Published,

実験手法

X-RAY DIFFRACTION (1.95 Å)