Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6BQD

TAF1-BD2 bromodomain in complex with (E)-3-(6-(but-2-en-1-yl)-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-N,N-dimethylbenzamide

Summary for 6BQD
Entry DOI10.2210/pdb6bqd/pdb
Related6BQA
DescriptorTranscription initiation factor TFIID subunit 1, 3-{6-[(2E)-but-2-en-1-yl]-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl}-N,N-dimethylbenzamide (3 entities in total)
Functional Keywordstaf1-bd2, bromodomain, gene regulation
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight30884.68
Authors
Murray, J.M.,Tang, Y. (deposition date: 2017-11-27, release date: 2019-02-20, Last modification date: 2023-10-04)
Primary citationNittinger, E.,Gibbons, P.,Eigenbrot, C.,Davies, D.R.,Maurer, B.,Yu, C.L.,Kiefer, J.R.,Kuglstatter, A.,Murray, J.,Ortwine, D.F.,Tang, Y.,Tsui, V.
Water molecules in protein-ligand interfaces. Evaluation of software tools and SAR comparison.
J. Comput. Aided Mol. Des., 33:307-330, 2019
Cited by
PubMed: 30756207
DOI: 10.1007/s10822-019-00187-y
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.136 Å)
Structure validation

217705

건을2024-03-27부터공개중

PDB statisticsPDBj update infoContact PDBjnumon