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6A93

Crystal structure of 5-HT2AR in complex with risperidone

Summary for 6A93
Entry DOI10.2210/pdb6a93/pdb
Descriptor5-hydroxytryptamine receptor 2A,Soluble cytochrome b562, 3-[2-[4-(6-fluoranyl-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one, CHOLESTEROL, ... (6 entities in total)
Functional Keywordsmembrane protein
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight86493.04
Authors
Kimura, T.K.,Asada, H.,Inoue, A.,Kadji, F.M.N.,Im, D.,Mori, C.,Arakawa, T.,Hirata, K.,Nomura, Y.,Nomura, N.,Aoki, J.,Iwata, S.,Shimamura, T. (deposition date: 2018-07-11, release date: 2019-02-13, Last modification date: 2023-11-22)
Primary citationKimura, K.T.,Asada, H.,Inoue, A.,Kadji, F.M.N.,Im, D.,Mori, C.,Arakawa, T.,Hirata, K.,Nomura, Y.,Nomura, N.,Aoki, J.,Iwata, S.,Shimamura, T.
Structures of the 5-HT2Areceptor in complex with the antipsychotics risperidone and zotepine.
Nat.Struct.Mol.Biol., 26:121-128, 2019
Cited by
PubMed: 30723326
DOI: 10.1038/s41594-018-0180-z
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3 Å)
Structure validation

217705

数据于2024-03-27公开中

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