6Z54
Crystal structure of CLK3 in complex with macrocycle ODS2003178
Summary for 6Z54
Entry DOI | 10.2210/pdb6z54/pdb |
Descriptor | Dual specificity protein kinase CLK3, 1,2-ETHANEDIOL, PHOSPHATE ION, ... (5 entities in total) |
Functional Keywords | kinase, kinase inhibitor, clk3, macrocycle, nanocyclic, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 43698.81 |
Authors | Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2020-05-26, release date: 2020-06-03, Last modification date: 2024-01-24) |
Primary citation | Chaikuad, A.,Benderitter, P.,Hoflack, J.,Denis, A.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of CLK3 in complex with macrocycle ODS2003178 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.73 Å) |
Structure validation
Download full validation report