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6GU2

CDK1/CyclinB/Cks2 in complex with Flavopiridol

Summary for 6GU2
Entry DOI10.2210/pdb6gu2/pdb
DescriptorCyclin-dependent kinase 1, G2/mitotic-specific cyclin-B1, Cyclin-dependent kinases regulatory subunit 2, ... (5 entities in total)
Functional Keywordscdk1, cyclinb1, cks2, inhibitor, cell cycle
Biological sourceHomo sapiens (Human)
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Total number of polymer chains3
Total formula weight76616.22
Authors
Wood, D.J.,Korolchuk, S.,Tatum, N.J.,Wang, L.Z.,Endicott, J.A.,Noble, M.E.M.,Martin, M.P. (deposition date: 2018-06-19, release date: 2018-12-05, Last modification date: 2024-01-17)
Primary citationWood, D.J.,Korolchuk, S.,Tatum, N.J.,Wang, L.Z.,Endicott, J.A.,Noble, M.E.M.,Martin, M.P.
Differences in the Conformational Energy Landscape of CDK1 and CDK2 Suggest a Mechanism for Achieving Selective CDK Inhibition.
Cell Chem Biol, 26:121-130.e5, 2019
Cited by
PubMed: 30472117
DOI: 10.1016/j.chembiol.2018.10.015
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

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