5Z9Q
Bacterial GyrB ATPase domain in complex with a chemical fragment
Summary for 5Z9Q
Entry DOI | 10.2210/pdb5z9q/pdb |
Descriptor | DNA gyrase subunit B, PHOSPHATE ION, 5-phenyl-1H-pyrazol-3-amine, ... (5 entities in total) |
Functional Keywords | dna topoisomerase, antibacterial, drug target, fragment-base lead discovery, isomerase |
Biological source | Escherichia coli (strain K12) |
Total number of polymer chains | 2 |
Total formula weight | 46242.36 |
Authors | |
Primary citation | Huang, X.,Guo, J.,Liu, Q.,Gu, Q.,Xu, J.,Zhou, H. Identification of an auxiliary druggable pocket in the DNA gyrase ATPase domain using fragment probes Medchemcomm, 9:1619-1629, 2018 Cited by PubMed: 30429968DOI: 10.1039/c8md00148k PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
Download full validation report