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5Z8G

BRD4 Bromodomain 1 with an inhibitor

Summary for 5Z8G
Entry DOI10.2210/pdb5z8g/pdb
DescriptorBromodomain-containing protein 4, 1-ethyl-6-[(3R)-3-oxidanylpiperidin-1-yl]sulfonyl-benzo[cd]indol-2-one, DIMETHYL SULFOXIDE, ... (4 entities in total)
Functional Keywordsbrd4 bromodomain 1, inhibitor, complex, transcription-inhibitor complex, transcription/inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15537.94
Authors
Xiao, S.,Chen, S.,Chen, H. (deposition date: 2018-01-31, release date: 2019-02-06, Last modification date: 2024-03-27)
Primary citationXiao, S.,Chen, S.,Chen, H.
BRD4 Bromodomain 1 with an inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.701 Å)
Structure validation

217705

건을2024-03-27부터공개중

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