5XY1
Crystal structure of Lyn kinase domain in complex with N-(1H-indazol-6-yl)-8-(piperidin-4-yloxy)-6-propylquinazolin-2-amine
Summary for 5XY1
Entry DOI | 10.2210/pdb5xy1/pdb |
Descriptor | Tyrosine-protein kinase Lyn, N-(1H-indazol-6-yl)-8-piperidin-4-yloxy-6-propyl-quinazolin-2-amine (3 entities in total) |
Functional Keywords | kinase, transferase |
Biological source | Homo sapiens (Human) |
Cellular location | Cell membrane: P07948 |
Total number of polymer chains | 1 |
Total formula weight | 32200.03 |
Authors | Kim, H.T. (deposition date: 2017-07-05, release date: 2017-08-02, Last modification date: 2023-11-22) |
Primary citation | Kim, H.T. Crystal structure of Lyn kinase domain in complex with N-(1H-indazol-6-yl)-8-(piperidin-4-yloxy)-6-propylquinazolin-2-amine To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
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