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5XI4

BRD4 bound with compound Bdi4

Summary for 5XI4
Entry DOI10.2210/pdb5xi4/pdb
DescriptorBromodomain-containing protein 4, (3~{S})-4-cyclopropyl-1,3-dimethyl-6-[[(1~{S})-1-(4-methylphenyl)ethyl]amino]-3~{H}-quinoxalin-2-one (3 entities in total)
Functional Keywordschromatin regulator, transcription-inhibitor complex, transcription/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains1
Total formula weight15103.54
Authors
Xiong, B.,Cao, D.,Li, Y. (deposition date: 2017-04-25, release date: 2018-05-02, Last modification date: 2024-03-27)
Primary citationXiong, B.,Cao, D.,Li, Y.
BRD4 bound with compound Bdi4
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.486 Å)
Structure validation

218500

數據於2024-04-17公開中

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