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5TCZ

NMR solution structure of engineered Protoxin-II analog

Summary for 5TCZ
Entry DOI10.2210/pdb5tcz/pdb
NMR InformationBMRB: 30181
DescriptorBeta/omega-theraphotoxin-Tp2a (1 entity in total)
Functional Keywordsvenom peptide analog, inhibitor, cystine knot, toxin
Biological sourceThrixopelma pruriens (Peruvian green velvet tarantula)
Total number of polymer chains1
Total formula weight3862.72
Authors
Gibbs, A.C.,Wickenden, A.D. (deposition date: 2016-09-16, release date: 2017-01-18)
Primary citationFlinspach, M.,Xu, Q.,Piekarz, A.D.,Fellows, R.,Hagan, R.,Gibbs, A.,Liu, Y.,Neff, R.A.,Freedman, J.,Eckert, W.A.,Zhou, M.,Bonesteel, R.,Pennington, M.W.,Eddinger, K.A.,Yaksh, T.L.,Hunter, M.,Swanson, R.V.,Wickenden, A.D.
Insensitivity to pain induced by a potent selective closed-state Nav1.7 inhibitor.
Sci Rep, 7:39662-39662, 2017
Cited by
PubMed: 28045073
DOI: 10.1038/srep39662
PDB entries with the same primary citation
Experimental method
SOLUTION NMR
Structure validation

217705

數據於2024-03-27公開中

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