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5TBH

Crystal structure of mouse CARM1 in complex with inhibitor LH1236

Summary for 5TBH
Entry DOI10.2210/pdb5tbh/pdb
DescriptorHistone-arginine methyltransferase CARM1, 1-METHOXY-2-(2-METHOXYETHOXY)ETHANE, 1,2-ETHANEDIOL, ... (7 entities in total)
Functional Keywordsprotein arginine methyltransferase, catalytic domain, chromatin regulator, mrna processing, mrna splicing, nucleus, s-adenosyl-l-methionine, transcription, transcription regulation, transferase
Biological sourceMus musculus (Mouse)
Total number of polymer chains4
Total formula weight166625.27
Authors
Cura, V.,Marechal, N.,Troffer-Charlier, N.,Halby, L.,Arimondo, P.,Bonnefond, L.,Cavarelli, J. (deposition date: 2016-09-12, release date: 2017-09-20, Last modification date: 2024-01-17)
Primary citationHalby, L.,Marechal, N.,Pechalrieu, D.,Cura, V.,Franchini, D.M.,Faux, C.,Alby, F.,Troffer-Charlier, N.,Kudithipudi, S.,Jeltsch, A.,Aouadi, W.,Decroly, E.,Guillemot, J.C.,Page, P.,Ferroud, C.,Bonnefond, L.,Guianvarc'h, D.,Cavarelli, J.,Arimondo, P.B.
Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors.
Philos.Trans.R.Soc.Lond.B Biol.Sci., 373:-, 2018
Cited by
PubMed: 29685976
DOI: 10.1098/rstb.2017.0072
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.341 Å)
Structure validation

217705

數據於2024-03-27公開中

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