5S5L
Tubulin-Z1492796719-complex
Summary for 5S5L
Entry DOI | 10.2210/pdb5s5l/pdb |
Group deposition | XChem fragment screening on T2R-TTL (G_1002173) |
Descriptor | Tubulin alpha-1B chain, N-[(3S)-1,2,3,4-tetrahydroquinolin-3-yl]acetamide, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... (12 entities in total) |
Functional Keywords | cell cycle, tubulin fold, cytoskeleton, microtubule |
Biological source | Rattus norvegicus (Rat) More |
Total number of polymer chains | 6 |
Total formula weight | 264736.61 |
Authors | Muehlethaler, T.,Gioia, D.,Prota, A.E.,Sharpe, M.E.,Cavalli, A.,Steinmetz, M.O. (deposition date: 2020-11-08, release date: 2021-06-30, Last modification date: 2024-03-06) |
Primary citation | Muhlethaler, T.,Gioia, D.,Prota, A.E.,Sharpe, M.E.,Cavalli, A.,Steinmetz, M.O. Comprehensive Analysis of Binding Sites in Tubulin. Angew.Chem.Int.Ed.Engl., 60:13331-13342, 2021 Cited by PubMed: 33951246DOI: 10.1002/anie.202100273 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.25 Å) |
Structure validation
Download full validation report