5O5U
X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a urea based inhibitor PSMA 1027
Summary for 5O5U
Entry DOI | 10.2210/pdb5o5u/pdb |
Descriptor | Glutamate carboxypeptidase 2, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (10 entities in total) |
Functional Keywords | glutamate carboxypeptidase ii (gcpii); naaladase; prostate-specific membrane antigen; urea based inhibitor, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 84636.62 |
Authors | Novakova, Z.,Barinka, C.,Motlova, L. (deposition date: 2017-06-02, release date: 2018-06-13, Last modification date: 2024-01-17) |
Primary citation | Novakova, Z.,Barinka, C.,Motlova, L. X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a urea based inhibitor PSMA 1027 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.53 Å) |
Structure validation
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