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5N84

TTK kinase domain in complex with Mps-BAY2b

Summary for 5N84
Entry DOI10.2210/pdb5n84/pdb
Related5N7V
DescriptorDual specificity protein kinase TTK, ~{N}-cyclopropyl-4-[8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide, SODIUM ION, ... (5 entities in total)
Functional Keywordskinase, inhibitor, mitosis, mps1, joost uitdehaag and nicole seegers 13021, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight36715.83
Authors
Uitdehaag, J.,Willemsen-Seegers, N.,de Man, J.,Buijsman, R.C.,Zaman, G.J.R. (deposition date: 2017-02-22, release date: 2017-05-31, Last modification date: 2024-01-17)
Primary citationUitdehaag, J.C.M.,de Man, J.,Willemsen-Seegers, N.,Prinsen, M.B.W.,Libouban, M.A.A.,Sterrenburg, J.G.,de Wit, J.J.P.,de Vetter, J.R.F.,de Roos, J.A.D.M.,Buijsman, R.C.,Zaman, G.J.R.
Target Residence Time-Guided Optimization on TTK Kinase Results in Inhibitors with Potent Anti-Proliferative Activity.
J. Mol. Biol., 429:2211-2230, 2017
Cited by
PubMed: 28539250
DOI: 10.1016/j.jmb.2017.05.014
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

217705

건을2024-03-27부터공개중

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