5JMY
NEPRILYSIN COMPLEXED WITH LBQ657
Summary for 5JMY
Entry DOI | 10.2210/pdb5jmy/pdb |
Descriptor | Neprilysin, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total) |
Functional Keywords | hydrolase, lbq657, sacubitril, heart failure |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 162585.10 |
Authors | Schiering, N.,Wiesmann, C. (deposition date: 2016-04-29, release date: 2016-06-15, Last modification date: 2024-01-10) |
Primary citation | Schiering, N.,D'Arcy, A.,Villard, F.,Ramage, P.,Logel, C.,Cumin, F.,Ksander, G.M.,Wiesmann, C.,Karki, R.G.,Mogi, M. Structure of neprilysin in complex with the active metabolite of sacubitril. Sci Rep, 6:27909-27909, 2016 Cited by PubMed: 27302413DOI: 10.1038/srep27909 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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