5ISO
STRUCTURE OF FULL LENGTH HUMAN AMPK (NON-PHOSPHORYLATED AT T-LOOP) IN COMPLEX WITH A SMALL MOLECULE ACTIVATOR, A BENZIMIDAZOLE DERIVATIVE (991)
Summary for 5ISO
Entry DOI | 10.2210/pdb5iso/pdb |
Descriptor | 5'-AMP-activated protein kinase catalytic subunit alpha-2, 5'-AMP-activated protein kinase subunit beta-1, 5'-AMP-activated protein kinase subunit gamma-1, ... (7 entities in total) |
Functional Keywords | transferase, nucleotide-binding, activator, non-phosphorylation |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 6 |
Total formula weight | 268846.82 |
Authors | Xiao, B.,Hubbard, J.A.,Gamblin, S.J. (deposition date: 2016-03-15, release date: 2017-03-29, Last modification date: 2024-01-10) |
Primary citation | Xiao, B.,Hubbard, J.A.,Gamblin, S.J. STRUCTURE OF FULL LENGTH HUMAN AMPK (NON-PHOSPHORYLATED AT T-LOOP) IN COMPLEX WITH A SMALL MOLECULE ACTIVATOR, A BENZIMIDAZOLE DERIVATIVE (991) To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.63 Å) |
Structure validation
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