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5IS9

Crystal structure of mouse CARM1 in complex with inhibitor SA0375

Summary for 5IS9
Entry DOI10.2210/pdb5is9/pdb
DescriptorHistone-arginine methyltransferase CARM1, (2S)-2-amino-4-[(3-{4-[(2S)-2-amino-2-carboxyethyl]-1H-1,2,3-triazol-1-yl}propyl){[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl}amino]butanoic acid (non-preferred name), 1,2-ETHANEDIOL, ... (8 entities in total)
Functional Keywordsprotein arginine methyltransferase, catalytic domain, chromatin regulator, mrna processing, mrna splicing, nucleus, s-adenosyl-l-methionine, transcription, transcription regulation, transferase
Biological sourceMus musculus (Mouse)
Cellular locationNucleus: Q9WVG6
Total number of polymer chains4
Total formula weight167582.31
Authors
Cura, V.,Marechal, N.,Mailliot, J.,Troffer-Charlier, N.,Hassenboehler, P.,Wurtz, J.M.,Bonnefond, L.,Cavarelli, J. (deposition date: 2016-03-15, release date: 2017-03-15, Last modification date: 2024-01-10)
Primary citationCura, V.,Marechal, N.,Mailliot, J.,Troffer-Charlier, N.,Wurtz, J.M.,Bonnefond, L.,Cavarelli, J.
Crystal structure of mouse CARM1 in complex with inhibitor SA0375
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

217705

数据于2024-03-27公开中

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