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5EW9

Crystal Structure of Aurora A Kinase Domain Bound to MK-5108

Summary for 5EW9
Entry DOI10.2210/pdb5ew9/pdb
DescriptorAurora kinase A, 4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid (3 entities in total)
Functional Keywordstransferase, protein kinase, inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationCytoplasm, cytoskeleton, microtubule organizing center, centrosome : O14965
Total number of polymer chains1
Total formula weight31998.99
Authors
Shiau, A.K.,Motamedi, A. (deposition date: 2015-11-20, release date: 2016-01-20, Last modification date: 2023-09-27)
Primary citationde Groot, C.O.,Hsia, J.E.,Anzola, J.V.,Motamedi, A.,Yoon, M.,Wong, Y.L.,Jenkins, D.,Lee, H.J.,Martinez, M.B.,Davis, R.L.,Gahman, T.C.,Desai, A.,Shiau, A.K.
A Cell Biologist's Field Guide to Aurora Kinase Inhibitors.
Front Oncol, 5:285-285, 2015
Cited by
PubMed: 26732741
DOI: 10.3389/fonc.2015.00285
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.181 Å)
Structure validation

225158

数据于2024-09-18公开中

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