5CU8
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2B (BAZ2B) in complex with 2-Amino-6-chlorobenzothiazole (SGC - Diamond I04-1 fragment screening)
5CU8 の概要
エントリーDOI | 10.2210/pdb5cu8/pdb |
分子名称 | Bromodomain adjacent to zinc finger domain protein 2B, 6-chloro-1,3-benzothiazol-2-amine, 1,2-ETHANEDIOL, ... (4 entities in total) |
機能のキーワード | structural genomics, structural genomics consortium, sgc, transcription |
由来する生物種 | Homo sapiens (Human) |
細胞内の位置 | Nucleus : Q9UIF8 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 13863.80 |
構造登録者 | Bradley, A.,Pearce, N.,Krojer, T.,Ng, J.,Talon, R.,Vollmar, M.,Jose, B.,von Delft, F.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2015-07-24, 公開日: 2015-09-09) |
主引用文献 | Bradley, A.,Pearce, N.,Krojer, T.,Ng, J.,Talon, R.,Vollmar, M.,Jose, B.,von Delft, F.,Bountra, C.,Arrowsmith, C.H.,Edwards, A.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of the second bromodomain of bromodomain adjancent to zinc finger domain protein 2B (BAZ2B) in complex with 2-Amino-6-chlorobenzothiazole (SGC - Diamond I04-1 fragment screening) To be published, |
実験手法 | X-RAY DIFFRACTION (2.05 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード