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5CA0

Crystal structure of T2R-TTL-Lexibulin complex

Summary for 5CA0
Entry DOI10.2210/pdb5ca0/pdb
Related5C8Y 5CA1 5CB4
DescriptorTubulin alpha-1B chain, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 1-ethyl-3-[2-methoxy-4-(5-methyl-4-{[(1S)-1-(pyridin-3-yl)butyl]amino}pyrimidin-2-yl)phenyl]urea, ... (13 entities in total)
Functional Keywordsinhibitor, complex, tubulin, structural protein
Biological sourceRattus norvegicus (Rat)
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Cellular locationCytoplasm, cytoskeleton: Q2XVP4 F2Z5B2
Golgi apparatus : P63043
Total number of polymer chains6
Total formula weight265378.76
Authors
Wang, Y.,Yu, Y.,Chen, Q.,Yang, J. (deposition date: 2015-06-29, release date: 2015-11-04, Last modification date: 2024-03-20)
Primary citationWang, Y.,Zhang, H.,Gigant, B.,Yu, Y.,Wu, Y.,Chen, X.,Lai, Q.,Yang, Z.,Chen, Q.,Yang, J.
Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283:102-111, 2016
Cited by
PubMed: 26462166
DOI: 10.1111/febs.13555
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.501 Å)
Structure validation

217705

数据于2024-03-27公开中

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