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5AP3

Naturally Occurring Mutations in the MPS1 Gene Predispose Cells to Kinase Inhibitor Drug Resistance.

5AP3 の概要
エントリーDOI10.2210/pdb5ap3/pdb
関連するPDBエントリー5AP0 5AP1 5AP2 5AP4 5AP5 5AP6 5AP7
分子名称DUAL SPECIFICITY PROTEIN KINASE TTK, 2-(2-(2-(2-(2-(2-ETHOXYETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHANOL, 9-CYCLOPENTYL-2-[[2-METHOXY-4-[(1-METHYLPIPERIDIN-4-YL)OXY]-PHENYL]AMINO]-7-METHYL-7,9-DIHYDRO-8H-PURIN-8-ONE, ... (6 entities in total)
機能のキーワードtransferase, mps1, protein kinase, mitosis, drug resistance
由来する生物種HOMO SAPIENS (HUMAN)
タンパク質・核酸の鎖数1
化学式量合計38123.63
構造登録者
主引用文献Gurden, M.D.,Westwood, I.M.,Faisal, A.,Naud, S.,Cheung, K.J.,Mcandrew, C.,Wood, A.,Schmitt, J.,Boxall, K.,Mak, G.,Workman, P.,Burke, R.,Hoelder, S.,Blagg, J.,Van Montfort, R.L.M.,Linardopoulos, S.
Naturally Occurring Mutations in the Mps1 Gene Predispose Cells to Kinase Inhibitor Drug Resistance.
Cancer Res., 75:3340-, 2015
Cited by
PubMed: 26202014
DOI: 10.1158/0008-5472.CAN-14-3272
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2.7 Å)
構造検証レポート
Validation report summary of 5ap3
検証レポート(詳細版)ダウンロードをダウンロード

217705

件を2024-03-27に公開中

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