Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5Z90

BRD4 Bromodomain 1 with an inhibitor

Summary for 5Z90
Entry DOI10.2210/pdb5z90/pdb
DescriptorBromodomain-containing protein 4, 1-ethyl-6-pyrrolidin-1-ylsulfonyl-benzo[cd]indol-2-one (3 entities in total)
Functional Keywordsbrd4 bromodomain 1, inhibitor, complex, transcription-inhibitor complex, transcription/inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15429.78
Authors
Xiao, S.,Chen, S.,Chen, H. (deposition date: 2018-02-01, release date: 2019-02-06, Last modification date: 2024-03-27)
Primary citationXiao, S.,Chen, S.,Chen, H.
BRD4 Bromodomain 1 with an inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon