5Z8R
BRD4 Bromodomain 1 with an inhibitor
Summary for 5Z8R
Entry DOI | 10.2210/pdb5z8r/pdb |
Descriptor | Bromodomain-containing protein 4, 1-ethyl-6-[(3S)-3-oxidanylpiperidin-1-yl]sulfonyl-benzo[cd]indol-2-one (3 entities in total) |
Functional Keywords | brd4 bromodomain 1, inhibitor, complex, transcription-inhibitor complex, transcription/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15459.81 |
Authors | |
Primary citation | Xiao, S.,Chen, S.,Chen, H. BRD4 Bromodomain 1 with an inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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