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5XHY

BRD4 bound with compound Bdi1

Summary for 5XHY
Entry DOI10.2210/pdb5xhy/pdb
DescriptorBromodomain-containing protein 4, ~{N}-(4-cyclopropyl-1,3,3-trimethyl-2-oxidanylidene-quinoxalin-6-yl)-4-methyl-benzenesulfonamide (3 entities in total)
Functional Keywordschromatin regulator, transcription-inhibitor complex, transcription/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains1
Total formula weight15153.58
Authors
Xiong, B.,Cao, D.,Li, Y. (deposition date: 2017-04-25, release date: 2018-05-02, Last modification date: 2024-03-27)
Primary citationBing, X.
BRD4 bound with compound Bdi1
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.976 Å)
Structure validation

222415

PDB entries from 2024-07-10

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