5ISB
Crystal structure of mouse CARM1 in complex with inhibitor SA0435
Summary for 5ISB
Entry DOI | 10.2210/pdb5isb/pdb |
Descriptor | Histone-arginine methyltransferase CARM1, 5'-{[(3S)-3-amino-3-carboxypropyl][(1H-imidazol-4-yl)methyl]amino}-5'-deoxyadenosine, 1,2-ETHANEDIOL, ... (7 entities in total) |
Functional Keywords | protein arginine methyltransferase, catalytic domain, chromatin regulator, mrna processing, mrna splicing, nucleus, s-adenosyl-l-methionine, transcription, transcription regulation, transferase |
Biological source | Mus musculus (Mouse) |
Cellular location | Nucleus: Q9WVG6 |
Total number of polymer chains | 4 |
Total formula weight | 167255.95 |
Authors | Cura, V.,Marechal, N.,Mailliot, J.,Troffer-Charlier, N.,Hassenboehler, P.,Wurtz, J.M.,Bonnefond, L.,Cavarelli, J. (deposition date: 2016-03-15, release date: 2017-03-29, Last modification date: 2024-01-10) |
Primary citation | Cura, V.,Marechal, N.,Mailliot, J.,Troffer-Charlier, N.,Wurtz, J.M.,Bonnefond, L.,Cavarelli, J. Crystal structure of mouse CARM1 in complex with inhibitor SA0435 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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