5ADT
Crystal structure of human tankyrase 2 in complex with OD73
Summary for 5ADT
Entry DOI | 10.2210/pdb5adt/pdb |
Related | 5ADQ 5ADR 5ADS |
Descriptor | TANKYRASE-2, BICARBONATE ION, SULFATE ION, ... (7 entities in total) |
Functional Keywords | transferase, protein-ligand complex, diphtheria toxin like fold, adp- ribosylation, transferase-transferase inhibitor complex |
Biological source | HOMO SAPIENS (HUMAN) More |
Cellular location | Cytoplasm: Q9H2K2 Q9H2K2 |
Total number of polymer chains | 2 |
Total formula weight | 27991.08 |
Authors | Haikarainen, T.,Lehtio, L. (deposition date: 2015-08-24, release date: 2016-01-13, Last modification date: 2024-05-08) |
Primary citation | Haikarainen, T.,Waaler, J.,Ignatev, A.,Nkizinkiko, Y.,Venkannagari, H.,Obaji, E.,Krauss, S.,Lehtio, L. Development and Structural Analysis of Adenosine Site Binding Tankyrase Inhibitors. Bioorg.Med.Chem.Lett., 26:328-, 2016 Cited by PubMed: 26706174DOI: 10.1016/J.BMCL.2015.12.018 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.15 Å) |
Structure validation
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