4XX5
Structure of PI3K gamma in complex with an inhibitor
Summary for 4XX5
Entry DOI | 10.2210/pdb4xx5/pdb |
Descriptor | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, N-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide (3 entities in total) |
Functional Keywords | transferase, inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Cytoplasm : P48736 |
Total number of polymer chains | 1 |
Total formula weight | 111060.53 |
Authors | Collier, P.N.,Messersmith, D.,Le Tiran, A.,Bandarage, U.K.,Boucher, C.,Come, J.,Cottrell, K.M.,Damagnez, V.,Doran, J.D.,Griffith, J.P.,Khare-Pandit, S.,Krueger, E.B.,Ledeboer, M.W.,Ledford, B.,Liao, Y.,Mahajan, S.,Moody, C.S.,Wang, T.,Xu, J.,Aronov, A.M. (deposition date: 2015-01-29, release date: 2015-08-05, Last modification date: 2024-02-28) |
Primary citation | Collier, P.N.,Messersmith, D.,Le Tiran, A.,Bandarage, U.K.,Boucher, C.,Come, J.,Cottrell, K.M.,Damagnez, V.,Doran, J.D.,Griffith, J.P.,Khare-Pandit, S.,Krueger, E.B.,Ledeboer, M.W.,Ledford, B.,Liao, Y.,Mahajan, S.,Moody, C.S.,Wang, T.,Xu, J.,Aronov, A.M. Structure of PI3K gamma in complex with an inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.76 Å) |
Structure validation
Download full validation report